STADA Superdrol(Methasterone)For Bodybuilding CAS:3381-88-2
Superdrol, chemically known as Methasterone (2α,17α-dimethyl-5α-androst-3-one-17β-ol), emerged in the 1950s as a synthetic anabolic steroid derived from dihydrotestosterone (DHT). Initially shelved due to concerns over toxicity, it resurfaced in the early 2000s as a "prohormone," marketed under brands like Superdrol and Methadrol.
Introduction to Superdrol: History and Background
Superdrol, chemically known as Methasterone (2α,17α-dimethyl-5α-androst-3-one-17β-ol), emerged in the 1950s as a synthetic anabolic steroid derived from dihydrotestosterone (DHT). Initially shelved due to concerns over toxicity, it resurfaced in the early 2000s as a "prohormone," marketed under brands like Superdrol and Methadrol. Its reputation skyrocketed in bodybuilding circles for rapid muscle gains, but regulatory crackdowns led to its classification as a controlled substance in the U.S. by 2012. Despite this, it persists in underground markets, celebrated for efficacy but notorious for risks.
Chemical Structure and Pharmacology
Methasterone's structure includes two methyl groups at the 2α and 17α positions, enhancing oral bioavailability and resistance to hepatic breakdown. The 17α-alkylation allows it to survive first-pass metabolism, but this modification exacerbates liver strain. Unlike testosterone, Superdrol cannot aromatize into estrogen, eliminating water retention. Its DHT backbone prevents conversion to potent androgens like dihydrotestosterone, focusing effects on muscle tissue with minimal androgenic activity.
Distinctive Features
●Anabolic-to-Androgenic Ratio: Estimated at 400:20, Superdrol prioritizes muscle growth over androgenic effects like acne or hair loss.
●Hepatotoxicity: The 17α-methyl group stresses liver enzymes, necessitating short cycles.
●Non-Estrogenic: Avoids estrogenic side effects (e.g., gynecomastia), making it a "dry" compound ideal for lean mass.
●Rapid Action: Users report noticeable strength and size gains within weeks.
Applications in Bodybuilding
●Bulking Cycles: Despite its dry nature, Superdrol is used off-season for lean mass accrual, often stacked with injectables like testosterone for synergistic effects.
●Cutting Phases: Preserves muscle during caloric deficits, enhancing vascularity and definition.
●Performance Enhancement: Athletes exploit its quick strength boosts for competitive edges, though detectable metabolites pose doping risks.
Benefits: Beyond Muscle Growth
●Efficiency: Gains of 10–15 pounds in 4–6 weeks are common, attributed to nitrogen retention and glycogenolysis.
●Strength Surges: Enhanced ATP synthesis in muscles fuels explosive training sessions.
●Aesthetic Enhancement: Promotes a hardened, vascular physique without subcutaneous fluid.
●Minimal Androgenic Effects: Reduced risk of hair loss or prostate issues compared to other steroids.
Risks and Side Effects
●Hepatic Stress: Elevated liver enzymes, jaundice, or hepatitis with prolonged use.
●Cardiovascular Strain: Alters lipid profiles, lowering HDL and raising LDL cholesterol.
●Endocrine Suppression: Shuts down natural testosterone production, necessitating PCT.
●General Toxicity: Reports of appetite loss, lethargy, and joint pain due to dry joints.
Dosage and Administration
●Beginners: 10–20 mg/day split into two doses (8–12 hours apart).
●Advanced Users: Up to 30 mg/day, though toxicity risks escalate.
●Cycle Duration: Strictly 4–6 weeks; extending use amplifies liver damage.
●Support Supplements: NAC (N-acetylcysteine) and TUDCA are employed to mitigate hepatic stress.
Half-Life and Timing
With a half-life of 8–12 hours, twice-daily dosing maintains stable blood levels. Morning and evening administration ensures sustained anabolic activity, though timing around workouts is debated for performance benefits.
Post-Cycle Therapy (PCT)
Post-cycle, users face suppressed natural testosterone. A 4–6 week PCT protocol includes:
●SERMs: Tamoxifen (20–40 mg/day) or Clomid (50–100 mg/day) to stimulate gonadotropins.
●HCG: Optional, to revive testicular function pre-PCT.
●Blood Work: Essential to monitor liver recovery and hormonal balance.
Legal Status and Accessibility
Classified as Schedule III in the U.S. and banned globally, Superdrol is illicit without a prescription. Black market products risk contamination or underdosing. Legal alternatives (e.g., DHEA-based products) mimic effects mildly but lack potency.
User Experiences and Community Perspectives
Anecdotes highlight polarized outcomes:
●Positive: Rapid gains, enhanced confidence, and competition-ready physiques.
●Negative: Hospitalizations from liver failure, post-cycle crashes, and long-term endocrine disruption.
Forums often warn newcomers of its "double-edged" nature, advocating reserved use for seasoned athletes.
Clinical data
|
Brand |
STADA |
|
Trade names |
Methyldrostanolone; Methasteron |
|
CAS |
3381-88-2 |
|
Molar mass |
318.501 |
|
Formula |
C21H34O2 |
|
Purity |
Above 98% |
|
Apprarance |
10mg*50 |
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Conclusion: Balancing Risk and Reward
Superdrol's allure lies in its unmatched efficiency for lean mass, yet its hepatotoxicity and legal risks demand caution. While it bypasses estrogenic pitfalls, the toll on hepatic and cardiovascular health underscores why medical professionals condemn its use. For bodybuilders weighing aesthetics against longevity, Superdrol remains a contentious choice-a testament to the sport's complex relationship with performance enhancement.
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